BA 1 TFA
产品介绍 | BA 1 TFA 是一种 bombesin (BB) 受体家族激动剂。BA 1 与 Bombesin 受体亚型 3 (BRS3),胃泌素释放肽受体 (GRPR),神经调节素 B 受体 (NMBR) 高亲和力结合,IC50 分别为 6、0.4、2.5 nM 。 | ||||||
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生物活性 | BA 1 TFA is a potent agonist for the bombesin (BB) family of receptors. BA1 binds with high affinity to Bombesin receptor subtype-3 (BRS3), gastrin releasing peptide receptor (GRPR), neuromedin B receptor (NMBR) with IC50s of 6, 0.4, 2.5 nM. | ||||||
体外研究 |
BA1 (0.1 μM) significantly increases FAK tyrosine phosphorylation in BRS-3 transfected NCI-H1299 cells. 西域 has not independently confirmed the accuracy of these methods. They are for reference only. | ||||||
体内研究 | |||||||
体内研究 | |||||||
性状 | Solid | ||||||
溶解性数据 | |||||||
运输条件 | Room temperature in continental US; may vary elsewhere. | ||||||
储存方式 |
Sealed storage, away from moisture and light
*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light) | ||||||
参考文献 |