DN02|西域试剂

DN02,99.17%

产品编号：Bellancom-148116| 分子式：C₂₂H₂₄FN₃O₃| 分子量：397.44

本网站销售的所有产品仅用于工业应用或者科学研究等非医疗目的,不可用于人类或动物的临床诊断或者治疗,非药用,非食用，

货号	包装	价格	库存与货期	购买量	操作
Bellancom-148116		￥4500.00	杭州北京（现货）
Bellancom-148116		￥8000.00	杭州北京（现货）

增值税发票√顺丰快递√订货电话：18601927057

DN02

产品介绍

DN02 是一种有效的选择性 BRD8 溴域探针。DN02 对 BRD8 (1) (K_i=32 nM) 具有较高的亲和力, 其亲和力是BRD8 (2) 的 30 倍 (K_i＞1000 nM)。

生物活性

DN02 is a potent, selective BRD8 bromodomain probe. DN02 has exhibits high affinity for the BRD8(1) (K_i=32 nM), which is 30-fold more affinity than BRD8 (2) (K_i＞1000 nM).

体外研究

DN02 has (1 nM-100 μM) low nM AlphaScreen with IC₅₀ value of 48 nM, with high selectivity over BRD9 and BRD4 in biochemical AlphaScreen assays.
DN02 (32 nM) has minimal off-target engagement across the bromodomain family, with modest activity against CBP/P300.

西域 has not independently confirmed the accuracy of these methods. They are for reference only.

体内研究

性状

Solid

溶解性数据

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式