Mal-NH-Boc|cas:134272-63-2|西域试剂

Mal-NH-Boc

产品编号：Bellancom-140991| CAS NO：134272-63-2| 分子式：C₁₁H₁₆N₂O₄| 分子量：240.26

Mal-NH-Boc 是一种 PROTAC linker，属于 alkyl/ether 类。可用于合成 PROTAC 分子。

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货号	包装	价格	库存与货期	购买量	操作
Bellancom-140991		￥210.00	杭州北京（现货）
Bellancom-140991		￥385.00	杭州北京（现货）

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Mal-NH-Boc

产品介绍

Mal-NH-Boc 是一种 PROTAC linker，属于 alkyl/ether 类。可用于合成 PROTAC 分子。

生物活性

Mal-NH-Boc is an alkyl/ether-based PROTAC linker that can be used in the synthesis of PROTACs.

体外研究

PROTACs contain two different ligands connected by a linker; one is a ligand for an E3 ubiquitin ligase and the other is for the target protein. PROTACs exploit the intracellular ubiquitin-proteasome system to selectively degrade target proteins.

西域 has not independently confirmed the accuracy of these methods. They are for reference only.

体内研究

性状

Solid

溶解性数据

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Powder	-20°C	3 years
	4°C	2 years
In solvent	-80°C	6 months
	-20°C	1 month

参考文献

. An S, et al. Small-molecule PROTACs: An emerging and promising approach for the development of targeted therapy drugs. EBioMedicine. 2018 Oct;36:553-562 [Content Brief]

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[1]. An S, et al. Small-molecule PROTACs: An emerging and promising approach for the development of targeted therapy drugs. EBioMedicine. 2018 Oct;36:553-562

Mal-NH-Boc

Mal-NH-Boc

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