Hydroxypropylmethyl cellulose acetate succinate (Mw: 20-100k Da),95.0%
产品编号:Bellancom-152927| CAS NO:71138-97-1| 分子式:| 分子量:
羟丙基甲基纤维素乙酸酯琥珀酸酯(Mw:20-100kDa)是制备低溶解度药物SDD的共溶剂。乙酸羟丙基甲基纤维素琥珀酸酯(Mw:20-100k Da)对大鼠无急性/亚慢性/慢性毒性,口服活性和LD50>2.5 g/kg。
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Hydroxypropylmethyl cellulose acetate succinate (Mw: 20-100k Da)
产品介绍 | Hydroxypropylmethyl cellulose acetate succinate (Mw: 20-100k Da) 是制备低溶解度活性分子 SDD 的助溶剂。Hydroxypropylmethyl cellulose acetate succinate (Mw: 20-100k Da) 口服有效,对大鼠无急性/亚慢性/慢性毒性,LD50 >2.5 g/kg。 | |||||||||
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生物活性 | Hydroxypropylmethyl cellulose acetate succinate (Mw: 20-100k Da) is a cosolvent for preparing SDDs of low-solubility agents. Hydroxypropylmethyl cellulose acetate succinate (Mw: 20-100k Da) exhibits no acute/subchronic/chronic toxicity in rats, with oral activity and LD50 >2.5 g/kg. | |||||||||
体外研究 | ||||||||||
体内研究 |
Hydroxypropylmethyl cellulose acetate succinate(2.5 g/kg;p.o.;单剂量)在大鼠无显著急性毒性。 西域 has not independently confirmed the accuracy of these methods. They are for reference only. | |||||||||
体内研究 |
Hydroxypropylmethyl cellulose acetate succinate(2.5 g/kg;p.o.;单剂量)在大鼠无显著急性毒性。 西域 has not independently confirmed the accuracy of these methods. They are for reference only. | |||||||||
性状 | Solid | |||||||||
溶解性数据 |
In Vitro:
DMSO : 100 mg/mL (Need ultrasonic) In Vivo:
请根据您的实验动物和给药方式选择适当的溶解方案。以下溶解方案都请先按照 In Vitro 方式配制澄清的储备液,再依次添加助溶剂:
——为保证实验结果的可靠性,澄清的储备液可以根据储存条件,适当保存;体内实验的工作液,建议您现用现配,当天使用;
以下溶剂前显示的百
*以上所有助溶剂都可在 西域 网站选购。
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运输条件 | Room temperature in continental US; may vary elsewhere. | |||||||||
储存方式 |
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参考文献 |

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