Glemanserin MDL11939,98.0%
产品编号:Bellancom-101250| CAS NO:107703-78-6| 分子式:C20H25NO| 分子量:295.42
本网站销售的所有产品仅用于工业应用或者科学研究等非医疗目的,不可用于人类或动物的临床诊断或者治疗,非药用,非食用,
Glemanserin MDL11939
产品介绍 | Glemanserin (MDL11939) 是有效和选择性 5-HT2A 受体的拮抗剂,对大鼠 5-HT2A、兔 5-HT2A 和人 5-HT2A 受体的 Ki 分别为 2.89、0.54 和 2.5 nM。 | ||||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
生物活性 | Glemanserin (MDL11939) is a potent and selective antagonist for serotonin receptor 5-HT2A (Ki=2.89, 0.54 and 2.5 nM for rat 5-HT2A, rabbit 5-HT2A and human 5-HT2A, respectively). | ||||||||||||
体外研究 | |||||||||||||
体内研究 |
Glemanserin (MDL11939) suppresses the induced increase in locomotor activity, behavioral sensitization and withdrawal symptoms in male mice. 西域 has not independently confirmed the accuracy of these methods. They are for reference only. | ||||||||||||
体内研究 |
Glemanserin (MDL11939) suppresses the induced increase in locomotor activity, behavioral sensitization and withdrawal symptoms in male mice. 西域 has not independently confirmed the accuracy of these methods. They are for reference only. | ||||||||||||
性状 | Solid | ||||||||||||
溶解性数据 | |||||||||||||
运输条件 | Room temperature in continental US; may vary elsewhere. | ||||||||||||
储存方式 |
| ||||||||||||
参考文献 |