FATP1-IN-1|cas:1431945-95-7|西域试剂

FATP1-IN-1,99.41%

产品编号：Bellancom-141699| CAS NO：1431945-95-7| 分子式：C₁₈H₂₂FN₅OS| 分子量：375.46

本网站销售的所有产品仅用于工业应用或者科学研究等非医疗目的,不可用于人类或动物的临床诊断或者治疗,非药用,非食用，

货号	价格	库存与货期
Bellancom-141699	￥3000.00	杭州北京（现货）
Bellancom-141699	￥4800.00	杭州北京（现货）
Bellancom-141699	￥9500.00	杭州北京（现货）
Bellancom-141699	￥14500.00	杭州北京（现货）

增值税发票√顺丰快递√订货电话：18601927057

FATP1-IN-1

产品介绍

FATP1-IN-1 (compound 5k) 是一种脂肪酸转运蛋白 1 (FATP1) 抑制剂。FATP1-IN-1 抑制重组人或小鼠 FATP1 acyl-CoA 合成酶活性，IC₅₀ 值分别为 0.046 μM和 0.60 μM。

生物活性

FATP1-IN-1 (compound 5k) is a fatty acid transport protein 1 (FATP1) inhibitor. FATP1-IN-1 is an inhibition of recombinant human or mouse acyl-CoA synthetase activity of FATP1, with the IC₅₀ values of 0.046 μM or 0.60 μM, respectively.

体外研究

体内研究

FATP1-IN-1 (p.o.; 10 mg/kg) treatment shows the C_max, AUC and T_max were 5.5 μg/mL, 36 μg h/mL and 0.33 hours, respectively, and exceeds the mouse IC₅₀ value of 0.22 μM without considering plasma protein binding.

西域 has not independently confirmed the accuracy of these methods. They are for reference only.

Animal Model:	Mouse plasma
Dosage:	10 mg/kg
Administration:	P.o.
Result:	The C_max, AUC and T_max were 5.5 μg/mL, 36 μg h/mL and 0.33 hours, respectively.

体内研究

西域 has not independently confirmed the accuracy of these methods. They are for reference only.

Animal Model:	Mouse plasma
Dosage:	10 mg/kg
Administration:	P.o.
Result:	The C_max, AUC and T_max were 5.5 μg/mL, 36 μg h/mL and 0.33 hours, respectively.

性状

Solid

溶解性数据

In Vitro:

DMSO : 62.5 mg/mL (166.46 mM; Need ultrasonic)

配制储备液

浓度溶剂体积质量	1 mg	5 mg	10 mg

1 mM	2.6634 mL	13.3170 mL	26.6340 mL
5 mM	0.5327 mL	2.6634 mL	5.3268 mL
10 mM	0.2663 mL	1.3317 mL	2.6634 mL

请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液；一旦配成溶液，请分装保存，避免反复冻融造成的产品失效。
储备液的保存方式和期限：-80°C, 6 months; -20°C, 1 month。-80°C 储存时，请在 6 个月内使用，-20°C 储存时，请在 1 个月内使用。

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式