hGPR91 antagonist 1|cas:1314796-00-3|西域试剂

hGPR91 antagonist 1,98.71%

产品编号：Bellancom-126217| CAS NO：1314796-00-3| 分子式：C₃₁H₂₃F₄N₃O| 分子量：529.53

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货号	价格	库存与货期
Bellancom-126217	￥2600.00	杭州北京（现货）
Bellancom-126217	￥3800.00	杭州北京（现货）
Bellancom-126217	￥8000.00	杭州北京（现货）
Bellancom-126217	￥12800.00	杭州北京（现货）

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hGPR91 antagonist 1

产品介绍

HGPR91 antagonist 1 是一种有效的，选择性小分子 hGPR91 拮抗剂，IC₅₀ 为 7 μM。

生物活性

HGPR91 antagonist 1 is a potent and selective small molecule hGPR91 antagonist with an IC₅₀ of 7 μM.

体外研究

体内研究

HGPR91 antagonist 1 leads to 59, 76% inhibition of ΔMAP at 2, 4 hours and has shown rat plasma protein binding 99%. HGPR91 antagonist 1 has engaged the target under the in vivo condition. HGPR91 antagonist 1 has clearance (CL) of 0.2 nmol/min/mg of RLM.

西域 has not independently confirmed the accuracy of these methods. They are for reference only.

Animal Model:	Wistar rats
Dosage:	100 mg/kg
Administration:	I.p.; 2 and 4 hours
Result:	Led to 59 and 76% inhibition of ΔMAP at 2 and 4 hours.

体内研究

西域 has not independently confirmed the accuracy of these methods. They are for reference only.

Animal Model:	Wistar rats
Dosage:	100 mg/kg
Administration:	I.p.; 2 and 4 hours
Result:	Led to 59 and 76% inhibition of ΔMAP at 2 and 4 hours.

性状

Solid

溶解性数据

In Vitro:

DMSO : ≥ 125 mg/mL (236.06 mM)

* "≥" means soluble, but saturation unknown.

配制储备液

浓度溶剂体积质量	1 mg	5 mg	10 mg

1 mM	1.8885 mL	9.4423 mL	18.8847 mL
5 mM	0.3777 mL	1.8885 mL	3.7769 mL
10 mM	0.1888 mL	0.9442 mL	1.8885 mL

请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液；一旦配成溶液，请分装保存，避免反复冻融造成的产品失效。
储备液的保存方式和期限：-80°C, 6 months; -20°C, 1 month。-80°C 储存时，请在 6 个月内使用，-20°C 储存时，请在 1 个月内使用。

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式