Glucocorticoid receptor agonist-1,95.16%
产品编号:Bellancom-131974| CAS NO:2166375-82-0| 分子式:C35H39NO6| 分子量:569.69
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Glucocorticoid receptor agonist-1
产品介绍 | Glucocorticoid receptor agonist-1 是一种有效的选择性 glucocorticoid receptor 激动剂,IC50 为 2.8 nM。详细信息请参考专利文献 WO2017210471A1 中的化合物 41。 |
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生物活性 | Glucocorticoid receptor agonist-1 is a potent glucocorticoid receptor agonist with an IC50 of 2.8 nM extracted from patent WO2017210471A1, compound 41. |
体外研究 |
Glucocorticoid receptor agonist immunoconjugates are useful for treating autoimmune diseases such as, but not limited to, rheumatoid arthritis, juvenile idiopathic arthritis, psoriatic arthritis, ankylosing spondylitis, adult Crohn's disease, pediatric Crohn's disease, ulcerative colitis, plaque psoriasis, hidradenitis suppurativa, uveitis, Behcets disease, a spondyloarthropathy, or psoriasis. 西域 has not independently confirmed the accuracy of these methods. They are for reference only. |
体内研究 | |
体内研究 | |
性状 | Solid |
溶解性数据 | |
运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 |
4°C, protect from light *In solvent : -80°C, 6 months; -20°C, 1 month (protect from light) |
参考文献 |